BDBM7401 (2 Z,3 E)-6-Bromoindirubin-3 -oxime::(3E)-6-bromo-3-[3-(hydroxyamino)indol-2-ylidene]oxindole::6-bromo-3-[(2Z,3E)-3-(hydroxyimino)-2,3-dihydro-1H-indol-2-ylidene]-2,3-dihydro-1H-indol-2-one::6-bromoindirubin-3 -oxime::6BIO::CHEMBL409450::indirubin deriv. 7a

SMILES Brc1ccc2C(C(=O)Nc2c1)c1[nH]c2ccccc2c1N=O

InChI Key InChIKey=OLOJSTRISMGUEK-UHFFFAOYSA-N

Data  24 IC50  1 EC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 7401   

TargetCasein kinase I isoform alpha(Sus scrofa)
University Of Athens

Curated by ChEMBL
LigandPNGBDBM7401((2 Z,3 E)-6-Bromoindirubin-3 -oxime | (3E)-6-bromo...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of porcine brain CK1 using RRKHAAIGpSAYSITA as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed